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3D structures from the PDB for "Dual specificity mitogen-activated protein kinase kinase 1" AND "BDBM50391802"
(Proteins have >= 85% sequence identity and ligands are exact matches)


Seq IdentityJmol DisplayPDB Title
4LMN100%JmolCRYSTAL STRUCTURE OF MEK1 KINASE BOUND TO GDC0973
7JUY>99%JmolCRYSTAL STRUCTURE OF KSR1:MEK1 IN COMPLEX WITH AMP-PNP, AND ALLOSTERIC MEK INHIBITOR COBIMETINIB
7M0V>99%JmolCRYSTAL STRUCTURE OF THE BRAF:MEK1 KINASES IN COMPLEX WITH AMPPNP AND COBIMETINIB
4AN286%JmolCRYSTAL STRUCTURES OF HUMAN MEK1 WITH CARBOXAMIDE-BASED ALLOSTERIC INHIBITOR XL518 (GDC-0973), OR RELATED ANALOGS.